Endocrine Therapy for Breast Cancer Risk Reduction
Recommendations
Tamoxifen
- Should be discussed as an option to reduce the risk of invasive BC, specifically ER-positive BC, in premenopausal women who are >35 years of age with a 5-year projected absolute BC risk >1.66% or with LCIS. Risk reduction benefit continues for at least 10 years.
- Is not recommended for use in women with a history of deep vein thrombosis, pulmonary embolus, stroke, transient ischemic attack, or during prolonged immobilization.
- Is not recommended for women who are pregnant, women who may become pregnant, or nursing mothers.
- Is not recommended in combination with hormone therapy.
- Follow-up should include a timely workup of abnormal vaginal bleeding.
- Discussions with patients and health care providers should include both the risks and benefits of tamoxifen in the preventive setting.
- Dosage: 20 mg/day orally for 5 years.
Raloxifene
- Should be discussed as an option to reduce the risk of invasive BC, specifically ER-positive BC, in postmenopausal women who are >35 years of age with a 5-year projected absolute BC risk >1.66% or with LCIS.
- May be used longer than 5 years in women with osteoporosis, in whom BC risk reduction is a secondary benefit.
- Should not be used for BC risk reduction in premenopausal women.
- Is not recommended for use in women with a history of deep vein thrombosis, pulmonary embolus, stroke, or transient ischemic attack, or during prolonged immobilization.
- Discussions with patients and health care providers should include both the risks and benefits of raloxifene in the preventive setting.
- Dosage: 60 mg/day orally for 5 years.
Exemestane
- Should be discussed as an alternative to tamoxifen and/or raloxifene to reduce the risk of invasive BC, specifically ER-positive BC, in postmenopausal women = 35 years of age with a 5-yearprojected absolute BC risk = 1.66% or with LCIS or atypical hyperplasia.
- Should not be used for BC risk reduction in premenopausal women.
- Discussions with patients and health care providers should include both the risks and benefits of exemestane in the preventive setting
- Dosage: 25 mg/day orally for 5 years.
Anastrozole
- Anastrozole (1 mg/day orally for 5 years) should be discussed as an alternative to tamoxifen, raloxifene, or exemestane to reduce the risk of invasive BC in postmenopausal women at increased risk of developing BC.
- Women most likely to benefit from endocrine therapy are those with one of more of the following: a diagnosis of atypical (ductal or lobular) hyperplasia or LCIS, an estimated 5-year risk (NCI BCRAT) of at least 3%, a 10-year risk (IBIS/Tyrer-Cuzick Risk Calculator) of at least 5%, or a relative risk of at least four times the population risk for their age group if their age is 40 to 44 years or two times the population risk for their age group if their age is 45 to 69 years.
- Clinicians should not prescribe anastrozole, exemestane, or raloxifene for BC risk reduction in premenopausal women.
- Discussions between patients and health care providers should include both the benefits and risks of anastrozole along with the other approved drugs for risk reduction based on menopausal status.
- Prior to initiating an aromatase inhibitor, clinicians should evaluate patients for baseline fracture risk and measure bone mineral density. Multiple studies have reported an increased rate of bone loss in women treated with aromatase inhibitors. Clinicians should use anastrozole with caution in postmenopausal women with moderate bone mineral density loss, and if it is used, they should consider the use of bone-protective agents such as bisphosphonates and RANKL inhibitors. All patients receiving aromatase inhibitors should be encouraged to exercise regularly and take adequate calcium and vitamin D supplements. A history of osteoporosis and/or severe bone loss is a relative contraindication for the use of anastrozole. In IBIS-II, women with severe osteoporosis (T score < -4 or more than two vertebral fractures) were excluded. Other endocrine preventive therapies that do not reduce bone density, such as tamoxifen or raloxifene, are also available for this group of women.
- Clinicians should also inform women of the possibility of joint stiffness, arthralgias, vasomotor symptoms, hypertension, dry eyes, and vaginal dryness while taking anastrozole.
Recommendation Grading
Overview
Title
Use of Endocrine Therapy for Breast Cancer Risk Reduction
Authoring Organization
American Society of Clinical Oncology
Publication Month/Year
September 3, 2019
Last Updated Month/Year
October 2, 2024
Supplemental Implementation Tools
Document Type
Guideline
External Publication Status
Published
Country of Publication
US
Document Objectives
To update the ASCO guideline on pharmacologic interventions for breast cancer risk reduction and provide guidance on clinical issues that arise when deciding to use endocrine therapy for breast cancer risk reduction.
Target Patient Population
Women without a personal history of breast cancer who are at increased risk of developing the disease
Target Provider Population
Medical oncologists, surgical oncologists, gynecologists, primary care physicians, and general practitioners
PICO Questions
What is the role of anastrozole in reducing the risk of developing breast cancer in women not previously diagnosed with breast cancer?
Inclusion Criteria
Female, Adult, Older adult
Health Care Settings
Ambulatory, Outpatient
Intended Users
Nurse, nurse practitioner, physician, physician assistant
Scope
Management
Diseases/Conditions (MeSH)
D001941 - Breast Diseases
Keywords
breast cancer, risk reduction, endocrine therapy, Breast Cancer
Source Citation
DOI: 10.1200/JCO.19.01472 Journal of Clinical Oncology 37, no. 33 (November 20, 2019) 3152-3165.